| 1 | BRD2, BRD3, BRD4, BRDT
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| PFI-1, a highly selective protein interaction inhibitor, targeting BET Bromodomains.
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| Picaud S, Da Costa D, Thanasopoulou A, Filippakopoulos P, Fish PV, Philpott M, Fedorov O, Brennan P, Bunnage ME, Owen DR, Bradner JE, Taniere P, O'Sullivan B, Müller S, Schwaller J, Stankovic T, Knapp S.
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| Cancer Res. Jun 1;73(11):3336-46. doi: 10.1158/0008-5472.CAN-12-3292. Epub 2013 Apr 10 2013
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| 2 | BRD2, BRD3, BRD4, BRDT
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| Discovery and Characterization of Small Molecule Inhibitors of the BET Family Bromodomains.
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| Chung CW, Coste H, White JH, Mirguet O, Wilde J, Gosmini RL, Delves C, Magny SM, Woodward R, Hughes SA, Boursier EV, Flynn H, Bouillot AM, Bamborough P, Brusq JM, Gellibert FJ, Jones EJ, Riou AM, Homes P, Martin SL, Uings IJ, Toum J, Clément CA, Boullay AB, Grimley RL, Blandel FM, Prinjha RK, Lee K, Kirilovsky J, Nicodeme E.
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| J Med Chem 54(11):3827-3838. Epub 2011 May 13.
2011
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| 3 | BRD3, GATA1
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| Structural Basis and Specificity of Acetylated Transcription Factor GATA1 Recognition by BET Family Bromodomain Protein Brd3.
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| Gamsjaeger R, Webb SR, Lamonica JM, Billin A, Blobel GA, Mackay JP.
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| Mol Cell Biol 31(13):2632-40. Epub 2011 May 9.
2011
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| 4 | BRD3, GATA1
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| Bromodomain protein Brd3 associates with acetylated GATA1 to promote its chromatin occupancy at erythroid target genes.
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| Lamonica JM, Deng W, Kadauke S, Campbell AE, Gamsjaeger R, Wang H, Cheng Y, Billin AN, Hardison RC, Mackay JP, Blobel GA.
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| Proc Natl Acad Sci U S A 108(22):E159-68. Epub 2011 May 2.
2011
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| 5 | BRD2, BRD3, BRD4, BRDT
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| Selective inhibition of BET bromodomains.
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| Filippakopoulos P, Qi J, Picaud S, Shen Y, Smith WB, Fedorov O, Morse EM, Keates T, Hickman TT, Felletar I, Philpott M, Munro S, McKeown MR, Wang Y, Christie AL, West N, Cameron MJ, Schwartz B, Heightman TD, La Thangue N, French CA, Wiest O, Kung AL, Knapp S, Bradner JE.
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| Nature 468(7327):1067-73. Epub 2010 Sep 24.
2010
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| 6 | BRD2, BRD3, BRD4, BRDT
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| Structural implications for K5/K12-di-acetylated histone H4 recognition by the second bromodomain of BRD2.
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| Umehara T, Nakamura Y, Wakamori M, Ozato K, Yokoyama S, Padmanabhan B.
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| FEBS Lett 584(18):3901-8. Epub 2010 Aug 13.
2010
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| 7 | BRD2, BRD3
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| The double bromodomain proteins Brd2 and Brd3 couple histone acetylation to transcription.
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| LeRoy G, Rickards B, Flint SJ.
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| Mol Cell 30(1):51-60.
2008
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| 8 | BRD2, BRD3, BRD4, BRDT
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| Bromodomain testis-specific protein is expressed in mouse oocyte and evolves faster than its ubiquitously expressed paralogs BRD2, -3, and -4.
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| Paillisson A, Levasseur A, Gouret P, Callebaut I, Bontoux M, Pontarotti P, Monget P.
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| Genomics 89(2):215-23. Epub 2006 Oct 16. 2007
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| 9 | BRD3
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| Differentially expressed genes in endothelial differentiation.
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| Ishii H, Mimori K, Mori M, Vecchione A.
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| DNA Cell Biol 24(7):432-7. 2005
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| 10 | NUP214, BRD3, RALGDS, RPL7A, TSC1
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| Mapping ESTs to the TSC1 candidate interval by use of the 'Science 96' transcript map.
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| Wolfe J, Jeremiah S, Young J, Burley MW, Stewart H, McCulley M, Grant C, Naz K, Povey S.
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| Ann Hum Genet 61(Pt 5):401-9. 1997
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| 11 | BRD2, BRD3
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| Chromosomal localization, gene structure and transcription pattern of the ORFX gene, a homologue of the MHC-linked RING3 gene.
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| Thorpe KL, Gorman P, Thomas C, Sheer D, Trowsdale J, Beck S.
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| Gene 200(1-2):177-83. 1997
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| 12 | BRD2, BRD3, NLRP1
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| Phylogeny and structure of the RING3 gene.
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| Thorpe KL, Abdulla S, Kaufman J, Trowsdale J, Beck S.
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| Immunogenetics 44(5):391-6. No abstract available. 1996
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